CAS
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861038-72-4
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英文名称
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A2764 dihydrochloride
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纯度
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≥98%
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分子式
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C15H21Cl3N2O
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分子量
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351.70
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外观(性状)
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Light yellow to yellow Solid
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储存条件
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Powder:2-8℃,2 years;In solvent(母液):-20℃,1 month; -80℃,6 months
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溶解性
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Soluble in Water ≥7mg/mL;Soluble in DMSO ≥4mg/mL(Need ultrasonic)
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描述
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A2764 dihydrochloride 是 TRESK (K2P18.1) 的高选择性抑制剂。(A2764 dihydrochloride is a highly selective inhibitor of TRESK (K2P18.1), having certain inhibitory effect on TREK-1 and TALK-1.)
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靶点
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Potassium Channel(TRESK (K2P18.1))
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通路
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Membrane Transporter&Ion Channel
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规格
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5mg
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单位
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瓶
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