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CAS
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32854-75-4
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中文名称
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高乌甲素
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英文名称
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Lappaconitine
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别名
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(+)-Lappaconitine;
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纯度
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HPLC≥98%
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分子式
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C32H44N2O8
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分子量
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584.7
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外观（性状）
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Off-white to light yellow Solid
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储存条件
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Powder : 2-8℃, 2 years; In solvent(母液): -20℃, 1 month; -80℃, 6 months
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溶解性
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Soluble in DMSO ≥10mg/mL
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InChIKey
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NWBWCXBPKTTZNQ-MUVXNFNYSA-N
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InChI
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InChI=1S/C32H44N2O8/c1-6-34-16-29(42-28(36)18-9-7-8-10-21(18)33-17(2)35)12-11-25(40-4)31-23(29)14-20(26(31)34)30(37)15-22(39-3)19-13-24(31)32(30,38)27(19)41-5/h7-10,19-20,22-27,37-38H,6,11-16H2,1-5H3,(H,33,35)/t19-,20-,22+,23-,24+,25+,26?,27+,29-,30+,31+,32+/m1/s1
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PubChem CID
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5281279
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SMILES
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CO[C@@H]1C(C(N(CC)C2)C3C4)([C@@](C[C@@]5([H])[C@@H]6OC)([H])[C@@]6(O)[C@@]3(C[C@@H]5OC)O)[C@@]4([H])[C@@]2(OC(C(C=CC=C7)=C7NC(C)=O)=O)CC1
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描述
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(Lappaconitine is a natural diterpenoid alkaloid (DTA) that acts as a sodium channel blocker with a wide range of biological activities, including antiarrhythmic, anti-inflammatory, antioxidant, anticancer, etc.)
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靶点
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P2X Receptor;Sodium Channel
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通路
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Membrane Transporter&Ion Channel
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规格
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20mg 10mM*1mL in DMSO 50mg 100mg
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单位
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瓶
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